Isometheptene
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| Image:Isometheptene.png | |
| Isometheptene
| |
| Systematic (IUPAC) name | |
| N,6-dimethylhept-5-en-2-amine | |
| Identifiers | |
| CAS number | |
| ATC code | A03 |
| PubChem | |
| Chemical data | |
| Formula | C9H19N |
| Mol. mass | 141.254 g/mol |
| Pharmacokinetic data | |
| Bioavailability | ? |
| Metabolism | ? |
| Half life | ? |
| Excretion | ? |
| Therapeutic considerations | |
| Pregnancy cat. |
? |
| Legal status | |
| Routes | Oral |
Isometheptene (usually as isometheptene mucate) is a sympathomimetic amine sometimes used in the treatment of migraines and tension headaches due to its vasoconstricting properties, that is, it causes constriction (narrowing) of blood vessels (arteries and veins). Along with paracetamol and dichloralphenazone, it is one of the constituents of Amidrine.
Chemistry
Isometheptene is a monounsaturated aliphatic secondary amine.
Drugs for functional gastrointestinal disorders (A03) | |
|---|---|
| Drugs for functional bowel disorders | antimuscarinics: Mebeverine - Dicycloverine - Propantheline
papaverine and derivatives: Papaverine - Drotaverine - Moxaverine acting on serotonin receptors: 5-HT3 antagonists (Alosetron, Cilansetron) - 5HT4 agonists (Mosapride, Tegaserod) other: Diisopromine - Isometheptene - Phloroglucinol - Proglumide - Tridihexethyl |
| Belladonna and derivatives (antimuscarinics) | Atropine - Hyoscyamine - Butylscopolamine - Methylscopolamine |
| Propulsives | primarily dopamine antagonists (Metoclopramide/Bromopride, Domperidone, Alizapride) - serotonin agonists (Cisapride) - Clebopride |
Sympathomimetic amines (R01, A08 and others) |
|---|
Alpha-pyrrolidinopropiophenone • Aminorex • d-Amphetamine & l,d-Amphetamine • d-Methamphetamine & l-Methamphetamine • Benzylpiperazine • Cathinone • CFT • Chlorphentermine • Clobenzorex • Cocaine • Cyclopentamine • Desoxypipradrol • Diethylpropion • Ephedrine • 4-FMP • 4-MTA • Fencamfamine • Fenfluramine • Fenproporex • Mazindol • MDPV • 4-Methyl-aminorex • Methylone • Methylphenidate • Naphazoline • Pemoline • Phendimetrazine • Phenmetrazine • Phentermine • Phenylephrine • Pipradrol • Pseudoephedrine • Pyrovalerone • Sibutramine • Synephrine |
| See also amphetamines |
Acknowledgement and Attribution Regarding Sources of Content
Some of the initial content on this page may be incorporated in part from copyleft sources in the public domain including wikis such as Wikipedia and AskDrWiki. Drug information for patients came from the The National Library of Medicine. Infectious disease information may have come from the Centers for Disease Control (CDC). Differential Diagnoses are drawn from clinicians as well as an amalgamation of 3 sources: 1.The Disease Database; 2. Kahan, Scott, Smith, Ellen G. In A Page: Signs and Symptoms. Malden, Massachusetts: Blackwell Publishing, 2004:3; 3. Sailer, Christian, Wasner, Susanne. Differential Diagnosis Pocket. Hermosa Beach, CA: Borm Bruckmeir Publishing LLC, 2002:7 .
