Phenprocoumon

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Phenprocoumon
Systematic (IUPAC) name
2-hydroxy-3-(1-phenylpropyl)chromen-4-one
Identifiers
CAS number 435-97-2
ATC code B01AA04
PubChem 9908
DrugBank APRD00228
Chemical data
Formula C18H16O3 
Mol. mass 280.318 g/mol
Pharmacokinetic data
Bioavailability  ?
Protein binding 99%
Metabolism hepatic to inactive metabolites
Half life 5 to 6 days
Excretion  ?
Therapeutic considerations
Pregnancy cat.

?

Legal status
Routes  ?

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Phenprocoumon

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Editor-In-Chief: C. Michael Gibson, M.S., M.D. [1]

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Phenprocoumon is an anticoagulant, functioning as a Vitamin K antagonist. It is a derivative of coumarin and is also marketed under the brand name Marcoumar. It is a vitamin K antagonist that inhibits coagulation by blocking synthesis of coagulation factors II, VII, IX and X. It is used for the prophylaxis and treatment of thromboembolic disorders.

It is marketed as Marcoumar by Roche.

External links


Cost Effectiveness of Phenprocoumon

| group5 = Clinical Trials Involving Phenprocoumon | list5 = Ongoing Trials on Phenprocoumon at Clinical Trials.govTrial results on PhenprocoumonClinical Trials on Phenprocoumon at Google


| group6 = Guidelines / Policies / Government Resources (FDA/CDC) Regarding Phenprocoumon | list6 = US National Guidelines Clearinghouse on PhenprocoumonNICE Guidance on PhenprocoumonNHS PRODIGY GuidanceFDA on PhenprocoumonCDC on Phenprocoumon


| group7 = Textbook Information on Phenprocoumon | list7 = Books and Textbook Information on Phenprocoumon


| group8 = Pharmacology Resources on Phenprocoumon | list8 = AND (Dose)}} Dosing of PhenprocoumonAND (drug interactions)}} Drug interactions with PhenprocoumonAND (side effects)}} Side effects of PhenprocoumonAND (Allergy)}} Allergic reactions to PhenprocoumonAND (overdose)}} Overdose information on PhenprocoumonAND (carcinogenicity)}} Carcinogenicity information on PhenprocoumonAND (pregnancy)}} Phenprocoumon in pregnancyAND (pharmacokinetics)}} Pharmacokinetics of Phenprocoumon


| group9 = Genetics, Pharmacogenomics, and Proteinomics of Phenprocoumon | list9 = AND (pharmacogenomics)}} Genetics of PhenprocoumonAND (pharmacogenomics)}} Pharmacogenomics of PhenprocoumonAND (proteomics)}} Proteomics of Phenprocoumon


| group10 = Newstories on Phenprocoumon | list10 = Phenprocoumon in the newsBe alerted to news on PhenprocoumonNews trends on Phenprocoumon</small>


| group11 = Commentary on Phenprocoumon | list11 = Blogs on Phenprocoumon

| group12 = Patient Resources on Phenprocoumon | list12 = Patient resources on PhenprocoumonDiscussion groups on PhenprocoumonPatient Handouts on PhenprocoumonDirections to Hospitals Treating PhenprocoumonRisk calculators and risk factors for Phenprocoumon


| group13 = Healthcare Provider Resources on Phenprocoumon | list13 = Symptoms of PhenprocoumonCauses & Risk Factors for PhenprocoumonDiagnostic studies for PhenprocoumonTreatment of Phenprocoumon

| group14 = Continuing Medical Education (CME) Programs on Phenprocoumon | list14 = CME Programs on Phenprocoumon

| group15 = International Resources on Phenprocoumon | list15 = Phenprocoumon en EspanolPhenprocoumon en Francais

| group16 = Business Resources on Phenprocoumon | list16 = Phenprocoumon in the MarketplacePatents on Phenprocoumon

| group17 = Informatics Resources on Phenprocoumon | list17 = List of terms related to Phenprocoumon


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